SCHEMBL16554188

SCHEMBL16554188

O=C(Nc1nc2cccc(O)c2s1)c1c(F)ccc(O)c1F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 7/20 0.65
HSD17B2 P37059 7/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
CYP2C9 P11712 1/20 0.65
CYP2B6 P20813 1/20 0.65
CYP2C19 P33261 1/20 0.65
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
GAA P10253 1/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TOP1 P11387 2/20 0.44
HPGD P15428 1/20 0.44
PCSK9 Q8NBP7 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16554186 0.82 HSD17B1 (0.63) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29964 0.79 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL10736618 0.68 SMN1; SMN2 (0.68) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL6067936 0.68 NPC1 (0.68) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL30432 0.68 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL5091421 0.68 NPC1 (0.66) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL30323 0.67 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL19612120 0.66 TMPRSS4 (0.54) MEN1KMT2A
SCHEMBL19627241 0.66 KCNMA1 (0.52) MEN1KMT2ANPC1RAB9ALMNA
SCHEMBL17251813 0.66 NPC1 (0.55) HSD17B1HSD17B2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041470-A1 METHODS AND COMPOSITIONS FOR SELECTIVE AND TARGETED CANCER THERAPY Board Of Regents Of the University Of Texas System (US) 2016-07-13 EP disclosed
WO-2015035051-A1 METHODS AND COMPOSITIONS FOR SELECTIVE AND TARGETED CANCER THERAPY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-03-12 WO disclosed