SCHEMBL165769

SCHEMBL165769

O=C(OCCN1CCCCC1)OCCN1CCCCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
ALDH1A1 P00352 2/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
PSMB1 P20618 1/20 0.47
PSMB5 P28074 1/20 0.47
PSMB2 P49721 1/20 0.47
CYP1A2 P05177 3/20 0.47
MAPK1 P28482 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
BCHE P06276 2/20 0.46
CYP2D6 P10635 2/20 0.44
TSHR P16473 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP2C9 P11712 1/20 0.44
THPO P40225 1/20 0.44
CHRM2 P08172 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL167209 0.98 KMT2A (0.51) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL12014419 0.88 KMT2A (0.49) KMT2AMEN1HPGDNPSR1
SCHEMBL3294445 0.87 THRB (0.50) KMT2AMEN1ALDH1A1MAPTPSMB1
SCHEMBL16829927 0.87 CYP2D6 (0.57) ALDH1A1POLBMAPTL3MBTL1CYP1A2
SCHEMBL12014424 0.85 KMT2A (0.46) KMT2AMEN1NPSR1
SCHEMBL165770 0.84 KMT2A (0.53) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL64387 0.83 KMT2A (0.45) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL328570 0.83 KMT2A (0.51) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL14959640 0.83 KMT2A (0.51) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL5093580 0.83 L3MBTL1 (0.55) KMT2AMEN1ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9018197-B2 Tetradecahydro-1H-cyclopenta[a]phenanthrene compounds, compositions, and related methods of use SUZHOU NEUPHARMA CO. LTD. (CN) 2015-04-28 US claimed
CN-102656179-A Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA CO LTD 2012-09-05 CN claimed
WO-2012027957-A1 BUFALIN DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF SUZHOU NEUPHARMA CO., LTD. (CN) 2012-03-08 WO claimed
CN-102656179-B Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA Co.,Ltd. (CN) 2015-07-29 CN disclosed
US-9018197-B2 Tetradecahydro-1H-cyclopenta[a]phenanthrene compounds, compositions, and related methods of use SUZHOU NEUPHARMA CO. LTD. (CN) 2015-04-28 US disclosed
CN-102656179-A Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA CO LTD 2012-09-05 CN disclosed
WO-2012027957-A1 BUFALIN DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF SUZHOU NEUPHARMA CO., LTD. (CN) 2012-03-08 WO disclosed