SCHEMBL1658804

SCHEMBL1658804

Cc1ccc(NC(=O)c2ccccc2S(=O)(=O)C(F)(F)F)cc1[AsH2]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.48
POLB P06746 1/20 0.47
CYP1A2 P05177 1/20 0.46
ALDH1A1 P00352 4/20 0.46
LMNA P02545 1/20 0.46
RXFP1 Q9HBX9 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
HTR2A P28223 1/20 0.42
TSPO P30536 1/20 0.42
GPR183 P32249 1/20 0.42
APLNR P35414 1/20 0.42
APOB P04114 2/20 0.42
MTTP P55157 2/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97456 0.88 CFTR (0.49) BCAT2POLBCYP1A2ALDH1A1LMNA
SCHEMBL100511 0.82 RAB9A (0.56) POLBALDH1A1LMNASMN1; SMN2NPC1
SCHEMBL1658803 0.78 SMN1; SMN2 (0.51) RXFP1SMN1; SMN2NPC1RAB9AHTT
SCHEMBL18921204 0.71 ALDH1A1 (0.48) BCAT2ALDH1A1MAPTHTR2AKDM4E
SCHEMBL7224833 0.69 BCAT2 (0.77) BCAT2POLBCYP1A2ALDH1A1LMNA
SCHEMBL20303506 0.69 NPC1 (0.57) POLBCYP1A2ALDH1A1LMNASMN1; SMN2
SCHEMBL11558124 0.69 TERT (0.48) POLBALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL29042565 0.68 CA1 (0.63) POLBALDH1A1LMNANPC1MAPT
SCHEMBL1408452 0.68 PTGS1 (0.66) CYP1A2ALDH1A1LMNARXFP1SMN1; SMN2
SCHEMBL5900421 0.68 PTGS1 (0.63) CYP1A2ALDH1A1LMNARXFP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011513379-A 2011-04-28 JP claimed
EP-2254882-A2 INTERMEDIATES AND A PROCESS EMPLOYING THE INTERMEDIATES FOR THE PREPARATION OF (3-TRIFLUOROMETHYLSULFONYL)-N-[4-METHYL-3- (4-PYRIDIN-3-YL-PYRIMIDIN-2YLAMINO)-PHENYL]-BENZAMIDE Natco Pharma Limited (IN) 2010-12-01 EP claimed
WO-2009109866-A2 INTERMEDIATES AND A PROCESS EMPLOYING THE INTERMEDIATES FOR THE PREPARATION OF (3-TRIFLUOROMETHYLSULFONYL)-N-[4-METHYL-3- (4-PYRIDIN-3-YL-PYRIMIDIN-2YLAMINO)-PHENYL]-BENZAMIDE NATCO PHARMA LIMITED (IN) 2009-09-11 WO claimed