SCHEMBL16588239

SCHEMBL16588239

C=CC[C@H](CCN(C(=O)OC)[C@@H](C)c1ccc(Br)cc1)c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.35
ROCK1 Q13464 1/20 0.33
CYP2C19 P33261 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ALDH1A1 P00352 2/20 0.32
PYCR1 P32322 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TXNRD1 Q16881 1/20 0.31
HTT P42858 2/20 0.31
MAPT P10636 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
CACNA1G O43497 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13538484 0.88 ALOX5 (0.37) ALOX5ROCK1CYP2C19PYCR1TRPM8
SCHEMBL13010741 0.79 CACNA1G (0.35) ALOX5ROCK1CACNA1G
SCHEMBL3655071 0.79 KMT2A (0.39) ALOX5SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL13077090 0.79 SLC6A4 (0.42) ALOX5SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL15959054 0.79 EPHX2 (0.34) ROCK1ALDH1A1TRPM8
SCHEMBL3655073 0.79 KMT2A (0.39) ALOX5SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL18380908 0.79 ALOX5 (0.35) ALOX5ROCK1SLC6A2SLC6A3ALDH1A1
SCHEMBL15436313 0.78 CYP2C19 (0.40) ALOX5CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL13538362 0.78 CYP2C19 (0.40) ALOX5CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL13552270 0.78 TRPM8 (0.34) ROCK1CYP2C19ALDH1A1NPSR1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220052-B1 CYCLIC UREA INHIBITORS OF 11ß-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS INC (US) 2015-03-25 EP disclosed