SCHEMBL16596227

SCHEMBL16596227

CCC(C)C(=O)Nc1ccnc(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.52
KCNB1 Q14721 1/20 0.49
SORT1 Q99523 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA14 Q9ULX7 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CNR1 P21554 1/20 0.42
ROCK2 O75116 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19308468 0.85 KCNB1 (0.56) KCNB1SORT1NPC1RAB9AKCNK3
SCHEMBL14920872 0.84 SORT1 (0.48) KCNB1SORT1KCNK3KCNK9ALDH1A1
SCHEMBL16596235 0.81 SMARCA2 (0.52) HSD17B10SORT1CA1CA2CA7
SCHEMBL18626324 0.80 SMARCA2 (0.55) HSD17B10CA1CA2CA7CA14
SCHEMBL16596226 0.80 HSD17B10 (0.48) HSD17B10CA1CA2CA7CA14
SCHEMBL19151039 0.80 KMT2A (0.53) SORT1RAB9AKCNK3KCNK9KDM4E
SCHEMBL19116521 0.79 MTNR1B (0.52) SORT1NPC1RAB9AKCNK3KCNK9
SCHEMBL15880285 0.77 SORT1 (0.55) SORT1KCNK3KCNK9ALDH1A1KMT2A
SCHEMBL13036336 0.77 SORT1 (0.52) HSD17B10SORT1NPC1RAB9AKCNK3
SCHEMBL19154013 0.77 MTNR1B (0.56) SORT1NPC1RAB9AKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015042363-A1 MOLECULES AND COMPOSITIONS THAT INHIBIT GRAM NEGATIVE BACTERIA AND THEIR USES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2015-03-26 WO disclosed