SCHEMBL16596235

SCHEMBL16596235

CCC(C)C(=O)Nc1ccnc(C)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.52
SMARCA4 P51532 1/20 0.52
PSEN1 P49768 6/20 0.49
PSEN2 P49810 6/20 0.49
APH1B Q8WW43 6/20 0.49
NCSTN Q92542 6/20 0.49
APH1A Q96BI3 6/20 0.49
PSENEN Q9NZ42 6/20 0.49
HSD17B10 Q99714 2/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA14 Q9ULX7 1/20 0.48
SORT1 Q99523 2/20 0.47
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.43
KDM4E B2RXH2 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16252564 0.84 SMARCA2 (0.58) SMARCA2SMARCA4PSEN1PSEN2APH1B
SCHEMBL18626324 0.84 SMARCA2 (0.55) SMARCA2SMARCA4HSD17B10CA1CA2
SCHEMBL16596226 0.84 HSD17B10 (0.48) HSD17B10CA1CA2CA7CA14
SCHEMBL16596227 0.81 HSD17B10 (0.52) HSD17B10CA1CA2CA7CA14
SCHEMBL16596228 0.80 SMARCA2 (0.54) SMARCA2SMARCA4CA1CA2CA7
SCHEMBL13134416 0.79 LMNA (0.60) HSD17B10CA1CA2CA7CA14
SCHEMBL18899922 0.78 SMARCA2 (0.58) SMARCA2SMARCA4SORT1LMNATSHR
SCHEMBL19116340 0.77 PTPN1 (0.54) SMARCA2SMARCA4SORT1LMNATSHR
SCHEMBL15880685 0.77 SMARCA2 (0.65) SMARCA2SMARCA4PSEN1PSEN2APH1B
SCHEMBL1949535 0.76 HSD17B10 (0.69) HSD17B10CA1CA2CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015042363-A1 MOLECULES AND COMPOSITIONS THAT INHIBIT GRAM NEGATIVE BACTERIA AND THEIR USES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2015-03-26 WO disclosed