SCHEMBL16601585

SCHEMBL16601585

Cc1ccc2c(c1)OCC(=O)N2C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.45
TSHR P16473 2/20 0.45
TERT O14746 1/20 0.44
PLK1 P53350 1/20 0.42
MMP12 P39900 1/20 0.40
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
GAA P10253 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3R1 P27986 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13340948 0.83 MAOB (0.38) HTTTSHRPOLBMAPTHSD17B10
SCHEMBL30921780 0.83 PIK3CD (0.46) CYP3A4CYP2D6MEN1KMT2AGAA
SCHEMBL14615641 0.83 SLC5A1 (0.43) HTTTERTMAPTHSD17B10PIK3CD
SCHEMBL13962148 0.83 CYP11B2 (0.36) HTTTSHRCYP2D6CYP11B1CYP11B2
SCHEMBL15798686 0.80 HTT (0.48) HTTTSHRPLK1CYP3A4CYP2D6
SCHEMBL7350158 0.79 ALOX12 (0.47) TSHRCYP2D6CYP2C19POLBMEN1
SCHEMBL5985192 0.79 CYP11B2 (0.55) HTTTSHRTERTPLK1MMP12
SCHEMBL18937271 0.79 TERT (0.48) HTTTERTCYP3A4CYP2C19CYP1A2
SCHEMBL8039853 0.76 SMN1; SMN2 (0.44) HTTPOLBALDH1A1MAPTHSD17B10
SCHEMBL18937270 0.76 MAPT (0.47) HTTTSHRCYP2C19CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993585-B2 Cyclic amine substituted pyrimidinediamines as PKC inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-03-31 US disclosed