SCHEMBL16601599

SCHEMBL16601599

Cc1ccc2c(c1)OCC(C(=O)N1CCN(C)CC1)O2

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
HPGD P15428 2/20 0.54
KMT2A Q03164 4/20 0.54
TP53 P04637 2/20 0.53
MAPT P10636 1/20 0.53
POLB P06746 3/20 0.52
MAPK1 P28482 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
TSHR P16473 1/20 0.52
GAA P10253 3/20 0.50
CYP3A4 P08684 1/20 0.50
ALOX12 P18054 1/20 0.50
CYP2C19 P33261 1/20 0.50
NPC1 O15118 1/20 0.48
THRB P10828 1/20 0.48
LMNA P02545 2/20 0.48
AIMP2 Q13155 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13962145 0.86 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2HPGDKMT2ATP53
SCHEMBL13341114 0.84 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2HPGDKMT2ATP53
SCHEMBL13202892 0.84 ALDH1A1 (0.76) ALDH1A1SMN1; SMN2HPGDKMT2APOLB
SCHEMBL15724692 0.82 HPGD (0.52) ALDH1A1SMN1; SMN2HPGDKMT2ATP53
SCHEMBL7437345 0.79 RAB9A (0.50) ALDH1A1SMN1; SMN2HPGDMAPTPOLB
SCHEMBL2054548 0.78 RAB9A (0.49) ALDH1A1SMN1; SMN2MAPTPOLBNPC1
SCHEMBL16601605 0.78 RAB9A (0.49) ALDH1A1SMN1; SMN2HPGDKMT2AMAPT
SCHEMBL1519184 0.78 RAB9A (0.49) ALDH1A1SMN1; SMN2MAPTPOLBNPC1
SCHEMBL1107089 0.78 RAB9A (0.49) ALDH1A1SMN1; SMN2MAPTPOLBNPC1
SCHEMBL9259044 0.75 KMT2A (0.61) ALDH1A1SMN1; SMN2HPGDKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993585-B2 Cyclic amine substituted pyrimidinediamines as PKC inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-03-31 US disclosed