SCHEMBL16610370

SCHEMBL16610370

COc1c(O)cc(C=O)cc1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
AOX1 Q06278 1/20 0.45
TDP1 Q9NUW8 2/20 0.41
TRIM24 O15164 2/20 0.41
TRIM33 Q9UPN9 2/20 0.41
HPGD P15428 1/20 0.41
ALDH5A1 P51649 1/20 0.41
ABAT P80404 1/20 0.41
APP P05067 2/20 0.40
TMPRSS4 Q9NRS4 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
TUBB1 Q9H4B7 1/20 0.36
KDM4E B2RXH2 2/20 0.36
PTGS2 P35354 1/20 0.36
RAB9A P51151 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KIF11 P52732 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL660556 0.88 KIF11 (0.40) ALDH1A1AOX1TDP1TRIM24TRIM33
SCHEMBL16610423 0.83 ALDH1A1 (0.45) ALDH1A1AOX1APPTUBB1KDM4E
SCHEMBL5155052 0.82 ALDH1A1 (0.57) ALDH1A1AOX1TDP1TRIM24TRIM33
SCHEMBL16077415 0.81 SRC (0.45) ALDH1A1AOX1TDP1TRIM24TRIM33
SCHEMBL896271 0.81 ALDH1A1 (0.46) ALDH1A1AOX1TDP1TRIM24TRIM33
SCHEMBL16610372 0.80 KDM4E (0.55) ALDH1A1TDP1HPGDAPPCA1
SCHEMBL16610333 0.79 APP (0.36) ALDH1A1HPGDAPPKDM4E
SCHEMBL1159670 0.77 TUBB1 (0.49) ALDH1A1AOX1TDP1TRIM24TRIM33
SCHEMBL8848334 0.77 XDH (0.46) ALDH1A1AOX1APPKDM4EPTGS2
SCHEMBL1458171 0.77 ALDH1A1 (0.49) ALDH1A1AOX1TDP1TRIM24TRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed