SCHEMBL16611014

SCHEMBL16611014

Cc1ccc(S(=O)(=O)OC2CCC(O[Si](C)(C)C(C)(C)C)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.51
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 3/20 0.34
TSHR P16473 2/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 2/20 0.34
USP2 O75604 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ENPP3 O14638 2/20 0.33
ENPP1 P22413 2/20 0.33
ENPP2 Q13822 2/20 0.33
HTR6 P50406 1/20 0.33
ACHE P22303 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16611088 1.00 CYP2D6 (0.51) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL16611012 1.00 CYP2D6 (0.51) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL4196702 0.92 CYP2D6 (0.46) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL16720978 0.89 CYP2D6 (0.45) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL16720982 0.89 CYP2D6 (0.45) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL20594990 0.87 CYP2D6 (0.44) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL31657622 0.84 ACHE (0.39) CYP2D6KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL1133701 0.84 CYP2D6 (0.36) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL21760775 0.84 CYP2D6 (0.36) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL1845464 0.84 CYP2D6 (0.36) CYP2D6CYP1A2CYP3A4CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250270211-A1 COMPOUNDS FOR FGFR INHIBITION COGENT BIOSCIENCES, INC. 2025-08-28 US disclosed
US-12351581-B2 Compounds for FGFR inhibition COGENT BIOSCIENCES, INC. (US) 2025-07-08 US disclosed
WO-2025034912-A9 COMPOUNDS FOR FGFR INHIBITION COGENT BIOSCIENCES, INC. (US) 2025-04-24 WO disclosed
US-20250066352-A1 COMPOUNDS FOR FGFR INHIBITION COGENT BIOSCIENCES, INC. 2025-02-27 US disclosed
WO-2025034912-A2 COMPOUNDS FOR FGFR INHIBITION COGENT BIOSCIENCES, INC. (US) 2025-02-13 WO disclosed
US-11396503-B2 Sulfonyl substituted bicyclic compound which acts as ROR inhibitor CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2022-07-26 US disclosed
CN-111094267-B Sulfonyl-substituted bicyclic compounds as ROR gamma inhibitors 正大天晴药业集团股份有限公司 2022-06-14 CN disclosed
US-11247990-B1 Bicyclic fused pyridine compounds as inhibitors of TAM kinases ARRAY BIOPHARMA INC (US) 2022-02-15 US disclosed
EP-3689860-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUND WHICH ACTS AS ROR INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-08-05 EP disclosed
US-20200239454-A1 SULFONYL SUBSTITUTED BICYCLIC COMPOUND WHICH ACTS AS ROR INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2020-07-30 US disclosed
CN-111094267-A Sulfonyl-substituted bicyclic compounds as ROR gamma inhibitors 正大天晴药业集团股份有限公司 2020-05-01 CN disclosed
WO-2019113190-A1 BICYCLIC FUSED PYRIDINE COMPOUNDS AS INHIBITORS OF TAM KINASES ARRAY BIOPHARMA INC. (US) 2019-06-13 WO disclosed
US-20160251352-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2016-09-01 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-20150141406-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-05-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160251352-A1 HETEROCYCLIC COMPOUND JAK2, JAK1, STAT3 CYP2D6 3478/4885CYP1A2 3322/4885CYP3A4 3938/4885
US-20250066352-A1 COMPOUNDS FOR FGFR INHIBITION FGFR1, FGFR4, FGFR3 CYP2D6 3242/4885CYP1A2 2094/4885CYP3A4 1663/4885
US-20250270211-A1 COMPOUNDS FOR FGFR INHIBITION FGFR1, FGFR4, FGFR3 CYP2D6 3242/4885CYP1A2 2094/4885CYP3A4 1663/4885
US-20200239454-A1 SULFONYL SUBSTITUTED BICYCLIC COMPOUND WHICH ACTS AS ROR INHIBITOR RORC, RORA, RORB CYP2D6 1402/4885CYP1A2 614/4885CYP3A4 447/4885
US-20150141406-A1 HETEROCYCLIC COMPOUND JAK2, JAK1, STAT3 CYP2D6 3478/4885CYP1A2 3322/4885CYP3A4 3938/4885
US-12351581-B2 Compounds for FGFR inhibition FGFR1, FGFR4, FGFR3 CYP2D6 3242/4885CYP1A2 2094/4885CYP3A4 1663/4885
US-11247990-B1 Bicyclic fused pyridine compounds as inhibitors of TAM kinases MAP3K1, MAP3K3, MAP3K2 CYP2D6 3215/4885CYP1A2 2249/4885CYP3A4 2186/4885
US-11396503-B2 Sulfonyl substituted bicyclic compound which acts as ROR inhibitor RORC, RORA, RORB CYP2D6 1402/4885CYP1A2 614/4885CYP3A4 447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.