SCHEMBL16612771

SCHEMBL16612771

COc1ccc2c(CCn3cc(N)cn3)cn(C)c2c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.50
HCRTR2 O43614 3/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HTR6 P50406 3/20 0.45
ALDH1A1 P00352 3/20 0.43
NQO2 P16083 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
HCRTR1 O43613 1/20 0.41
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.37
HASPIN Q8TF76 1/20 0.37
SSTR5 P35346 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12479701 0.91 ADRB2 (0.63) ADRB2HCRTR2MEN1KMT2AHTR6
SCHEMBL12479868 0.80 HTR2A (0.57) HCRTR2MEN1KMT2AALDH1A1LMNA
SCHEMBL16612680 0.79 HTR2A (0.58) HCRTR2MEN1KMT2AHTR6MTNR1A
SCHEMBL2029351 0.78 ADRB2 (0.78) ADRB2MEN1KMT2AHTR6ALDH1A1
SCHEMBL12479182 0.77 HTR2A (0.58) HCRTR2MEN1KMT2AHTR6MTNR1A
SCHEMBL1703175 0.74 MEN1 (0.76) HCRTR2MEN1KMT2A
SCHEMBL13888163 0.73 ALDH1A1 (0.60) ADRB2MEN1KMT2AHTR6ALDH1A1
SCHEMBL10507566 0.73 ADRB2 (0.55) ADRB2MEN1KMT2AHTR6ALDH1A1
SCHEMBL25624145 0.73 HTR6 (0.80) ADRB2HTR6
SCHEMBL16612770 0.73 ADRB2 (0.44) ADRB2HCRTR2MEN1KMT2AHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed