SCHEMBL16612923

SCHEMBL16612923

NC(=O)c1[c]cn(CCOc2nc3ccccc3o2)n1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 8/20 0.43
KCNH2 Q12809 1/20 0.42
HCRTR2 O43614 2/20 0.40
HCRTR1 O43613 1/20 0.40
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CNR2 P34972 5/20 0.35
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612601 0.78 DDAH1 (0.50) NPC1RAB9AL3MBTL1SMN1; SMN2HPGD
SCHEMBL16612797 0.78 HCRTR2 (0.40) HCRTR2NPC1RAB9AL3MBTL1TP53
SCHEMBL16613039 0.78 MEN1 (0.46) HCRTR2HCRTR1NPC1RAB9AL3MBTL1
SCHEMBL16612643 0.77 HCRTR1 (0.39) HCRTR2HCRTR1L3MBTL1
SCHEMBL16613032 0.75 HCRTR2 (0.44) HCRTR2
SCHEMBL16612999 0.73 HCRTR2 (0.53) LTA4HKCNH2HCRTR2HCRTR1NPC1
SCHEMBL16612782 0.72 HCRTR2 (0.39) HCRTR2HCRTR1
SCHEMBL16612739 0.71 TDP1 (0.54) NPC1L3MBTL1SMN1; SMN2HPGD
SCHEMBL9403508 0.70 KMT2A (0.44) LTA4HNPC1RAB9AL3MBTL1TP53
SCHEMBL16612710 0.70 KDM4E (0.49) HCRTR2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed