SCHEMBL16612643

SCHEMBL16612643

NC(=O)c1[c]cn(CCOc2ncc3ccccc3n2)n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
POLB P06746 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
IKBKB O14920 1/20 0.31
SYK P43405 1/20 0.30
AURKB Q96GD4 1/20 0.30
CTDSP1 Q9GZU7 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16613039 0.81 MEN1 (0.46) HCRTR1HCRTR2POLBTDP1MEN1
SCHEMBL16612683 0.79 FDPS (0.45) HCRTR2SYK
SCHEMBL16612877 0.79 HCRTR2 (0.35) HCRTR2SYKAURKB
SCHEMBL16612923 0.77 LTA4H (0.43) HCRTR1HCRTR2L3MBTL1
SCHEMBL16612712 0.74 HCRTR2 (0.38) HCRTR1HCRTR2POLBTDP1
SCHEMBL16612710 0.73 KDM4E (0.49) HCRTR2POLBMEN1MAPTKMT2A
SCHEMBL16612782 0.73 HCRTR2 (0.39) HCRTR1HCRTR2
SCHEMBL16613011 0.71 HCRTR2 (0.36) HCRTR1HCRTR2
SCHEMBL16612850 0.71 HCRTR2 (0.38) HCRTR1HCRTR2MAPT
SCHEMBL16612857 0.70 MTNR1A (0.44) TDP1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed