SCHEMBL16615168

SCHEMBL16615168

O=C(c1c2c3c(n1-2)NCCN3Cc1c(Cl)ccc(F)c1Cl)N1CCN(c2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
HTT P42858 1/20 0.40
LMNA P02545 3/20 0.38
PKM P14618 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 5/20 0.38
REN P00797 2/20 0.38
CLEC4M Q9H2X3 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
HSP90AA1 P07900 1/20 0.37
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
TP53 P04637 1/20 0.36
MEN1 O00255 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615221 0.78 L3MBTL1 (0.40) LMNAALDH1A1PTGS2KDM4ETP53
SCHEMBL20859311 0.78 HTT (0.41) KMT2AHTTLMNAPKMNPSR1
SCHEMBL16615153 0.77 PLK4 (0.41) KMT2AHTTLMNAPKMNPSR1
SCHEMBL12146409 0.75 PLK4 (0.46) KMT2AHTTLMNAPKMNPSR1
SCHEMBL17969745 0.75 KDM4E (0.39) ALDH1A1KDM4EUSP2TSHR
SCHEMBL20859452 0.73 LMNA (0.35) KMT2AHTTLMNAPKMALDH1A1
SCHEMBL17969728 0.66 ALK (0.49)
SCHEMBL16615217 0.65 KCNQ2 (0.44) KMT2AHTTALDH1A1KDM4EMEN1
SCHEMBL16615279 0.64 HDAC1 (0.33)
SCHEMBL16615102 0.64 MAPT (0.44) KMT2AHTTLMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed