SCHEMBL16615186

SCHEMBL16615186

Clc1ccc(Cl)c(CN2CCNc3c2c2c(-c4nnc(C5CCNCC5)[nH]4)n3-2)c1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.34
BRAF P15056 1/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
GPR6 P46095 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615167 0.84 MAP4K3 (0.31)
SCHEMBL16615075 0.79 ALK (0.42) ALKBRAFSLC6A2SLC6A4NPC1
SCHEMBL16615324 0.78 ALK (0.34) ALK
SCHEMBL16615327 0.74 ALK (0.40) ALK
SCHEMBL16615077 0.73 BCHE (0.39) ALKSLC6A2SLC6A4GPR6
SCHEMBL16615265 0.72 NPC1 (0.43) ALKGPR6NPC1RAB9A
SCHEMBL16615266 0.71 LMNA (0.38) ALK
SCHEMBL20859278 0.71 ALK (0.33) ALKBRAFSLC6A2SLC6A4
SCHEMBL16615084 0.71 ALK (0.46) ALKBRAF
SCHEMBL16615336 0.70 LMNA (0.35) ALKNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed