SCHEMBL16615265

SCHEMBL16615265

Clc1ccc(Cl)c(CN2CCNc3c2c2c(-c4nc(C5CCCCC5)no4)n3-2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
POLB P06746 2/20 0.35
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALK Q9UM73 1/20 0.33
PDE2A O00408 1/20 0.33
HSD11B1 P28845 1/20 0.32
RXFP3 Q9NSD7 1/20 0.31
GPR6 P46095 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615276 0.88 ALK (0.32) CHRM1CHRM3ALKGPR6
SCHEMBL17918692 0.79 NPC1 (0.42) NPC1RAB9ASMN1; SMN2CHRM1CHRM3
SCHEMBL17969717 0.79 ALK (0.40) CHRM1CHRM3MEN1KMT2AKDM4E
SCHEMBL16615200 0.78 CHRM1 (0.45) NPC1RAB9ASMN1; SMN2CHRM1CHRM3
SCHEMBL16615327 0.76 ALK (0.40) ALDH1A1ALKKCNH2
SCHEMBL16615324 0.75 ALK (0.34) ALDH1A1ALKKCNH2
SCHEMBL16615266 0.75 LMNA (0.38) SMN1; SMN2ALDH1A1HPGDMEN1KMT2A
SCHEMBL16615336 0.74 LMNA (0.35) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL16615186 0.72 ALK (0.34) NPC1RAB9AALKGPR6
SCHEMBL17918690 0.68 ALK (0.40) NPC1RAB9ASMN1; SMN2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed