SCHEMBL16615327

SCHEMBL16615327

CN1CCC(c2nnc(-c3c4c5c(n3-4)NCCN5Cc3cc(Cl)ccc3Cl)o2)CC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.40
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
KCNH2 Q12809 1/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 2/20 0.35
ENPP2 Q13822 3/20 0.34
TNKS O95271 2/20 0.33
PARP1 P09874 2/20 0.33
PARP2 Q9UGN5 2/20 0.33
LRRK2 Q5S007 1/20 0.33
HTR4 Q13639 1/20 0.33
ALOX15B O15296 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615328 0.89 ALK (0.43) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615324 0.89 ALK (0.34) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615266 0.85 LMNA (0.38) ALKMAPTALDH1A1
SCHEMBL16615365 0.85 PLK4 (0.35) ALKDRD2DRD3KCNH2TP53
SCHEMBL17918694 0.79 ALK (0.49) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615265 0.76 NPC1 (0.43) ALKKCNH2ALDH1A1
SCHEMBL16615186 0.74 ALK (0.34) ALK
SCHEMBL16615276 0.73 ALK (0.32) ALKMAPT
SCHEMBL17969717 0.72 ALK (0.40) ALKLRRK2
SCHEMBL20859343 0.72 ALK (0.36) ALKDRD2DRD3KCNH2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed