SCHEMBL16615215

SCHEMBL16615215

O=C(Nc1cccc(C(=O)N2CCCC2)c1)c1c2c3c(n1-2)NCCN3Cc1cc(Cl)ccc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 5/20 0.50
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
TSHR P16473 1/20 0.38
TP53 P04637 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
EPHX2 P34913 2/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615216 0.86 ALK (0.49) ALK
SCHEMBL16615268 0.85 KDM4E (0.41) POLBKDM4EHTTRAB9ATP53
SCHEMBL17918802 0.81 ALK (0.60) ALKPOLBKDM4EHTTKMT2A
SCHEMBL17969783 0.77 ALK (0.48) ALKPOLBKDM4EHTTKMT2A
SCHEMBL16615217 0.77 KCNQ2 (0.44) POLBKDM4EHTTKMT2ANPC1
SCHEMBL16615358 0.76 CCNC (0.46) ALK
SCHEMBL16615299 0.74 POLB (0.41) ALKPOLBKMT2ANPC1RAB9A
SCHEMBL16615074 0.74 MAPT (0.45) POLBKDM4EHTTKMT2ANPC1
SCHEMBL20859453 0.72 ALK (0.43) ALKPOLBKDM4EHTTKMT2A
SCHEMBL16615305 0.72 KMT2A (0.40) POLBKDM4EHTTKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed