SCHEMBL16615358

SCHEMBL16615358

O=C(Nc1ccc(C(=O)N2CCNCC2)cc1)c1c2c3c(n1-2)NCCN3Cc1cc(Cl)ccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNC P24863 12/20 0.46
CDK8 P49336 12/20 0.46
MC4R P32245 1/20 0.40
MC5R P33032 1/20 0.40
MC3R P41968 1/20 0.40
MC1R Q01726 1/20 0.40
MAPT P10636 1/20 0.39
FLT3 P36888 1/20 0.38
ALK Q9UM73 1/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615299 0.92 POLB (0.41) CCNCCDK8MC5RMAPTFLT3
SCHEMBL16615074 0.92 MAPT (0.45) MAPTFLT3
SCHEMBL16615268 0.91 KDM4E (0.41) CCNCCDK8
SCHEMBL16615216 0.90 ALK (0.49) CCNCCDK8MC4RMC5RMC3R
SCHEMBL16615102 0.82 MAPT (0.44) MAPT
SCHEMBL17918724 0.79 CCNC (0.47) CCNCCDK8MAPTFLT3ALK
SCHEMBL16615217 0.78 KCNQ2 (0.44) MAPT
SCHEMBL16615213 0.76 EPHX2 (0.43) MAPTFLT3
SCHEMBL16615215 0.76 ALK (0.50) ALK
SCHEMBL20859294 0.75 CCNC (0.41) CCNCCDK8MC4RMC5RMC3R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed