SCHEMBL16615216

SCHEMBL16615216

O=C(Nc1ccc(C(=O)N2CCNCC2)cc1)c1c2c3c(n1-2)NCCN3Cc1cc(Cl)ccc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.49
CCNC P24863 8/20 0.43
CDK8 P49336 8/20 0.43
DDR1 Q08345 3/20 0.39
SLC2A1 P11166 1/20 0.38
MC4R P32245 1/20 0.36
MC5R P33032 1/20 0.36
MC3R P41968 1/20 0.36
MC1R Q01726 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615358 0.90 CCNC (0.46) ALKCCNCCDK8MC4RMC5R
SCHEMBL16615215 0.86 ALK (0.50) ALK
SCHEMBL16615074 0.82 MAPT (0.45)
SCHEMBL16615299 0.82 POLB (0.41) ALKCCNCCDK8MC5R
SCHEMBL16615268 0.81 KDM4E (0.41) CCNCCDK8
SCHEMBL16615213 0.75 EPHX2 (0.43)
SCHEMBL16615102 0.73 MAPT (0.44)
SCHEMBL17918724 0.70 CCNC (0.47) ALKCCNCCDK8
SCHEMBL16615217 0.69 KCNQ2 (0.44)
SCHEMBL17918802 0.68 ALK (0.60) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed