SCHEMBL16615283

SCHEMBL16615283

CNC1CCN(c2cccc(NC(=O)c3c4c5c(n3-4)NCCN5Cc3c(Cl)ccc(F)c3Cl)c2)CC1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SETD2 Q9BYW2 5/20 0.38
NSD2 O96028 1/20 0.38
ALDH1A1 P00352 4/20 0.37
MALT1 Q9UDY8 1/20 0.35
ACKR3 P25106 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.34
IDO1 P14902 1/20 0.34
ACHE P22303 1/20 0.34
HTR1A P08908 1/20 0.34
CNR1 P21554 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KCNQ2 O43526 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615218 0.82 SETD2 (0.37) SETD2NSD2ALDH1A1MALT1ACKR3
SCHEMBL16615217 0.78 KCNQ2 (0.44) ALDH1A1KDM4EMAPTCNR1KCNQ2
SCHEMBL17918850 0.73 SETD2 (0.48) SETD2NSD2MALT1ACKR3MAPT
SCHEMBL16615221 0.73 L3MBTL1 (0.40) ALDH1A1KDM4EMAPT
SCHEMBL20859460 0.69 SETD2 (0.46) SETD2NSD2MALT1ACKR3IDO1
SCHEMBL16615102 0.67 MAPT (0.44) ALDH1A1KDM4EMAPTTDP1
SCHEMBL16615268 0.67 KDM4E (0.41) KDM4E
SCHEMBL25037760 0.66 SETD2 (0.79) SETD2NSD2
SCHEMBL17969758 0.65 EGFR (0.39)
SCHEMBL16615305 0.65 KMT2A (0.40) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed