SCHEMBL16622225

SCHEMBL16622225

CC(=O)Nc1ccc(C#Cc2ccc(CC(N)=O)cc2)cn1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.46
ACACB O00763 14/20 0.44
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432897 0.87 RAB9A (0.44) PTK2ACACBRAB9AMEN1KMT2A
Hydrochloric Acid SCHEMBL1432991 0.86 RAB9A (0.43) PTK2ACACBRAB9AMEN1KMT2A
SCHEMBL16622218 0.86 ACACB (0.43) ACACBRAB9AMEN1KMT2AKDM4E
SCHEMBL27809191 0.81 ACACB (0.44) PTK2ACACBRAB9AMEN1KMT2A
SCHEMBL16622212 0.80 KMT2A (0.69) ACACBRAB9AMEN1KMT2AKDM4E
SCHEMBL16622220 0.80 EGLN1 (0.41) ACACBRAB9AMEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL27981821 0.80 ACACB (0.43) PTK2ACACBRAB9AMEN1KMT2A
SCHEMBL16622211 0.76 KDM4E (0.45) ACACBRAB9AMEN1KMT2AKDM4E
SCHEMBL1432507 0.75 ACACB (0.42) ACACBRAB9AMEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL1432946 0.74 ACACB (0.41) ACACBRAB9AMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999989-B2 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-TECH UENO, LTD. (JP) 2015-04-07 US disclosed