SCHEMBL16622218

SCHEMBL16622218

CC(=O)Nc1cnc(C#Cc2ccc(CC(N)=O)cc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACACB O00763 16/20 0.43
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432507 0.89 ACACB (0.42) ACACBKDM4EMEN1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL1432946 0.88 ACACB (0.41) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL16622225 0.86 PTK2 (0.46) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL27809002 0.83 ACACB (0.43) ACACBKDM4EMEN1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL27981776 0.82 ACACB (0.43) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL16622212 0.77 KMT2A (0.69) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL1432897 0.77 RAB9A (0.44) ACACBKDM4EMEN1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL1432991 0.76 RAB9A (0.43) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL16622220 0.75 EGLN1 (0.41) ACACBKDM4EMEN1ALDH1A1HPGD
SCHEMBL16622211 0.73 KDM4E (0.45) ACACBKDM4EMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999989-B2 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-TECH UENO, LTD. (JP) 2015-04-07 US disclosed