SCHEMBL16622219

SCHEMBL16622219

NC(=O)COc1ccc(C#Cc2ccc(CC(N)=O)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.51
LMNA P02545 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
CNR1 P21554 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
KDM4E B2RXH2 1/20 0.49
CYP1A2 P05177 1/20 0.49
GLA P06280 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
THPO P40225 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
CA2 P00918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1433216 0.86 ALDH1A1 (0.48) FFAR1LMNATDP1ADRB2ADRB1
Hydrochloric Acid SCHEMBL1432917 0.85 ALDH1A1 (0.47) FFAR1LMNATDP1ADRB2ADRB1
SCHEMBL23582957 0.81 ALOX15 (0.57) FFAR1CA2
SCHEMBL23582938 0.81 PLA2G4B (0.55) CA2
SCHEMBL10506137 0.80 MEN1 (0.58) TDP1KDM4EBLM
SCHEMBL9517796 0.79 POLB (0.54) LMNATDP1ADRB2ADRB1CNR1
SCHEMBL9450347 0.79 MEN1 (0.49) TDP1BLM
SCHEMBL16254218 0.79 FFAR1 (0.72) FFAR1CA2
SCHEMBL6539400 0.77 KMT2A (0.49) FFAR1TDP1KDM4EBLM
SCHEMBL3371954 0.77 MEN1 (0.51) TDP1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999989-B2 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-TECH UENO, LTD. (JP) 2015-04-07 US disclosed