SCHEMBL16623486

SCHEMBL16623486

N=C(c1ccc(CCNC2CC2)cc1)c1c(Nc2c(F)cccc2F)c(Br)c[nH]c1=O

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.32
RAB9A P51151 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623518 0.80 KMT2A (0.31)
SCHEMBL17849207 0.75 ROCK1 (0.39) RAB9A
SCHEMBL16726672 0.73 CDK2 (0.32)
SCHEMBL16623533 0.73 F10 (0.34)
SCHEMBL16726665 0.69 ALDH2 (0.33)
SCHEMBL16726670 0.69
SCHEMBL17849208 0.69 HDAC6 (0.33)
SCHEMBL16623450 0.69 NPC1 (0.32)
SCHEMBL17849189 0.68 RAB9A (0.45) RAB9A
SCHEMBL17849220 0.67 MT-CO2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed