SCHEMBL16623562

SCHEMBL16623562

N=C(c1cccc(CN)c1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.39
CFD P00746 3/20 0.32
EGFR P00533 1/20 0.32
ENPP2 Q13822 1/20 0.31
HTR2C P28335 1/20 0.31
ALDH2 P05091 1/20 0.31
F10 P00742 2/20 0.31
F11 P03951 1/20 0.31
TPSB2 P20231 1/20 0.31
SUCNR1 Q9BXA5 1/20 0.31
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623601 0.90 PRSS1 (0.37) EGFRALDH2PRSS1PRSS2PRSS3
SCHEMBL17849229 0.89 F10 (0.35) EGFRALDH2F10PRSS1PRSS2
SCHEMBL16623485 0.85 PARP1 (0.37) CDK8
SCHEMBL16623496 0.84 CYP2D6 (0.42) EGFR
SCHEMBL16623507 0.82 ITGA4 (0.33) EGFRF10
SCHEMBL16623511 0.80 TYK2 (0.38)
SCHEMBL16623603 0.80 PARP1 (0.36) ALDH2
SCHEMBL16623558 0.79 PARP1 (0.34)
SCHEMBL16623497 0.78 JAK2 (0.32) EGFR
SCHEMBL16726648 0.78 KDR (0.33) ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed