SCHEMBL16623507

SCHEMBL16623507

CCC(C)C(=O)Cc1cccc(C(=N)c2c(Nc3c(F)cccc3F)cc[nH]c2=O)c1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
F10 P00742 2/20 0.32
PTGS2 P35354 1/20 0.32
F2 P00734 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849229 0.85 F10 (0.35) F10PTGS2F2EGFR
SCHEMBL16623569 0.84 PTGS2 (0.31) PTGS2
SCHEMBL16623601 0.83 PRSS1 (0.37) PTGS2EGFR
SCHEMBL16623562 0.82 LOXL2 (0.39) F10EGFR
SCHEMBL16623485 0.78 PARP1 (0.37)
SCHEMBL16623496 0.77 CYP2D6 (0.42) EGFR
SCHEMBL16726656 0.75 PTGS2 (0.33) PTGS2
SCHEMBL16623511 0.73 TYK2 (0.38)
SCHEMBL17849242 0.73 PTGS2 (0.34) PTGS2EGFR
SCHEMBL16623603 0.73 PARP1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed