SCHEMBL16623496

SCHEMBL16623496

N=C(c1cccc(CN2CCCC2)c1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HIF1A Q16665 1/20 0.42
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EGFR P00533 1/20 0.36
CHRM3 P20309 1/20 0.35
PTPN2 P17706 1/20 0.35
IGF1R P08069 1/20 0.35
ACKR3 P25106 1/20 0.35
CACNA1G O43497 1/20 0.34
HTR3A P46098 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
PARP1 P09874 1/20 0.34
GLS O94925 1/20 0.34
NTRK1 P04629 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623601 0.85 PRSS1 (0.37) EGFR
SCHEMBL16623562 0.84 LOXL2 (0.39) EGFR
SCHEMBL17849229 0.82 F10 (0.35) EGFR
SCHEMBL16623485 0.78 PARP1 (0.37) PARP1
SCHEMBL17849238 0.78 L3MBTL1 (0.38) EGFRIGF1RPARP1NTRK1
SCHEMBL16623507 0.77 ITGA4 (0.33) EGFR
SCHEMBL16623503 0.75 EGFR (0.35) EGFRPARP1
SCHEMBL16623565 0.74 ALDH1A1 (0.41) CYP2D6CYP2C9ALDH1A1SMN1; SMN2
SCHEMBL16623558 0.74 PARP1 (0.34) PARP1
SCHEMBL17849249 0.74 EGFR (0.40) ALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed