SCHEMBL17849229

SCHEMBL17849229

N=C(c1cccc(CC(N)=O)c1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.35
PTGS2 P35354 2/20 0.34
EGFR P00533 2/20 0.32
ABCB11 O95342 1/20 0.32
PTGS1 P23219 1/20 0.32
PPARG P37231 1/20 0.32
NR1I3 Q14994 1/20 0.32
ALDH2 P05091 1/20 0.32
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31
F2 P00734 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16726656 0.90 PTGS2 (0.33) PTGS2ABCB11PTGS1PPARGNR1I3
SCHEMBL16623562 0.89 LOXL2 (0.39) F10EGFRALDH2PRSS1PRSS2
SCHEMBL16623601 0.88 PRSS1 (0.37) PTGS2EGFRALDH2PRSS1PRSS2
SCHEMBL17849242 0.87 PTGS2 (0.34) PTGS2EGFRABCB11PTGS1PPARG
SCHEMBL16623485 0.86 PARP1 (0.37)
SCHEMBL16623507 0.85 ITGA4 (0.33) F10PTGS2EGFRF2
SCHEMBL16623533 0.82 F10 (0.34) F10PRSS1PRSS2PRSS3
SCHEMBL16623511 0.82 TYK2 (0.38)
SCHEMBL16623496 0.82 CYP2D6 (0.42) EGFR
SCHEMBL16623603 0.81 PARP1 (0.36) ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed