SCHEMBL16623592

SCHEMBL16623592

Cc1c[nH]c(=O)c(C(=N)c2ccc(N3CCNC3=O)cc2)c1Nc1c(F)cccc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.35
CMA1 P23946 6/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
F10 P00742 1/20 0.32
HCRTR1 O43613 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGAV P06756 1/20 0.32
ITGA5 P08648 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB5 P18084 1/20 0.32
ITGB8 P26012 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
RORC P51449 1/20 0.32
ELANE P08246 2/20 0.32
TDO2 P48775 1/20 0.31
SCN9A Q15858 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623594 0.96 CMA1 (0.35) EIF2AK2CMA1NPC1RAB9AF10
SCHEMBL17849212 0.89 ITGB3 (0.37) EIF2AK2CMA1NPC1RAB9AF10
SCHEMBL17849219 0.84 RAF1 (0.42) NPC1RAB9AMEN1KMT2A
SCHEMBL17849221 0.83 EIF2AK2 (0.34) EIF2AK2CMA1NPC1RAB9AHCRTR1
SCHEMBL17849193 0.75 F10 (0.43) NPC1RAB9AF10LMNA
SCHEMBL16623554 0.75 MAPK14 (0.33) F10KMT2A
SCHEMBL16623479 0.74 CRBN (0.40) EIF2AK2CMA1
SCHEMBL16623587 0.73 ROCK1 (0.39) NPC1RAB9A
SCHEMBL16623480 0.73 MAPK14 (0.34) F10RORCKMT2A
SCHEMBL17849207 0.72 ROCK1 (0.39) NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed