SCHEMBL17849221

SCHEMBL17849221

N=C(c1ccc(N2CCNC2=O)cc1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.34
EGFR P00533 11/20 0.34
ITGB3 P05106 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA5 P08648 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB5 P18084 1/20 0.33
ITGB8 P26012 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SCN9A Q15858 1/20 0.32
PARP1 P09874 1/20 0.31
HCRTR1 O43613 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
RORC P51449 1/20 0.31
CMA1 P23946 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623503 0.86 EGFR (0.35) EGFRPARP1JAK2JAK1
SCHEMBL16623565 0.85 ALDH1A1 (0.41) NPC1RAB9A
SCHEMBL17849249 0.85 EGFR (0.40) EGFRJAK2JAK1
SCHEMBL18052623 0.85 EGFR (0.36) EGFRSCN9AJAK2JAK1RORC
SCHEMBL17849188 0.83 EGFR (0.40) EGFRNPC1RAB9AJAK2JAK1
SCHEMBL16623493 0.83 TYK2 (0.39) JAK2JAK1
SCHEMBL17849212 0.83 ITGB3 (0.37) EIF2AK2ITGB3ITGB1ITGAVITGA5
SCHEMBL16623592 0.83 EIF2AK2 (0.35) EIF2AK2ITGB3ITGB1ITGAVITGA5
SCHEMBL16623558 0.80 PARP1 (0.34) PARP1
SCHEMBL16623594 0.79 CMA1 (0.35) EIF2AK2ITGB3ITGB1ITGAVITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed