SCHEMBL16623479

SCHEMBL16623479

Cc1c[nH]c(=O)c(C(=N)c2ccc3c(c2)NC(=O)C3)c1Nc1c(F)cccc1F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 2/20 0.40
SMYD3 Q9H7B4 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
HDAC3 O15379 2/20 0.33
GRIA1 P42261 2/20 0.33
CACNG8 Q8WXS5 2/20 0.33
HDAC1 Q13547 1/20 0.33
EPHX2 P34913 1/20 0.33
CMA1 P23946 2/20 0.33
AHR P35869 2/20 0.33
EIF2AK2 P19525 1/20 0.32
MGLL Q99685 1/20 0.31
HSD11B1 P28845 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
TDP2 O95551 2/20 0.30
KIF11 P52732 1/20 0.30
KDR P35968 1/20 0.30
PLK1 P53350 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849215 0.90 CRBN (0.38) CRBNSMYD3HDAC3HDAC1EPHX2
SCHEMBL16623554 0.77 MAPK14 (0.33)
SCHEMBL16623480 0.75 MAPK14 (0.34) KDR
SCHEMBL17849219 0.75 RAF1 (0.42)
SCHEMBL16623552 0.73 DDB1 (0.32) CRBNBRD4CREBBP
SCHEMBL16623594 0.71 CMA1 (0.35) CMA1EIF2AK2
SCHEMBL17849205 0.69 DGAT1 (0.32)
SCHEMBL17849236 0.68 RORC (0.36)
SCHEMBL17849202 0.67 SMN1; SMN2 (0.44)
SCHEMBL17849213 0.67 POLB (0.35) HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed