SCHEMBL16623480

SCHEMBL16623480

Cc1c[nH]c(=O)c(C(=N)c2cc(C(N)=O)ccc2F)c1Nc1c(F)cccc1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.34
PDGFRB P09619 1/20 0.32
KDR P35968 1/20 0.32
RORC P51449 1/20 0.32
PARP1 P09874 5/20 0.32
KMT2A Q03164 1/20 0.31
F10 P00742 2/20 0.31
F2 P00734 1/20 0.31
PLG P00747 1/20 0.31
PLAU P00749 1/20 0.31
PLAT P00750 1/20 0.31
KLK1 P06870 1/20 0.31
KLK5 Q9Y337 1/20 0.31
ERN1 O75460 1/20 0.31
GUSB P08236 1/20 0.31
KAT6A Q92794 1/20 0.30
CHRM2 P08172 2/20 0.30
CHRM1 P11229 2/20 0.30
RRM1 P23921 2/20 0.30
RRM2B Q7LG56 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849237 0.89 RORC (0.33) MAPK14RORCPARP1GUSB
SCHEMBL16623554 0.86 MAPK14 (0.33) MAPK14KMT2AF10F2PLG
SCHEMBL16623600 0.82 TYK2 (0.34) MAPK14PARP1ERN1KAT6A
SCHEMBL16623479 0.75 CRBN (0.40) KDR
SCHEMBL17849205 0.75 DGAT1 (0.32) MAPK14F10GUSB
SCHEMBL17849236 0.74 RORC (0.36) MAPK14RORCPARP1KMT2A
SCHEMBL17849219 0.73 RAF1 (0.42) MAPK14KMT2A
SCHEMBL16623552 0.73 DDB1 (0.32)
SCHEMBL16623485 0.70 PARP1 (0.37) PARP1KMT2AERN1
SCHEMBL16623511 0.70 TYK2 (0.38) PARP1KAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed