SCHEMBL16624100

SCHEMBL16624100

CCN1CCc2c([nH]c3cc(C)ccc23)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.50
TRPV1 Q8NER1 1/20 0.49
ACHE P22303 4/20 0.48
GRIN1 Q05586 3/20 0.48
GRIN2A Q12879 3/20 0.48
GRIN2B Q13224 3/20 0.48
GRIN2D O15399 2/20 0.48
GRIN3B O60391 2/20 0.48
GRIN2C Q14957 2/20 0.48
GRIN3A Q8TCU5 2/20 0.48
DRD2 P14416 1/20 0.48
DRD1 P21728 1/20 0.48
DRD4 P21917 1/20 0.48
DRD5 P21918 1/20 0.48
SIGMAR1 Q99720 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ATM Q13315 2/20 0.44
GAA P10253 1/20 0.44
RCE1 Q9Y256 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17993875 0.85 MEN1 (0.55) HTR1ATRPV1GRIN2BDRD2DRD1
SCHEMBL17993840 0.83 HTR7 (0.55) HTR1ATRPV1ACHEDRD2DRD1
SCHEMBL6369610 0.81 HTR1A (0.71) HTR1AGRIN2BDRD2DRD1DRD4
SCHEMBL18034956 0.81 KDM4E (0.66) TRPV1ACHEGRIN1GRIN2AGRIN2B
SCHEMBL17993835 0.80 KDM4E (0.46) TRPV1ACHEGRIN1GRIN2AGRIN2B
SCHEMBL25512896 0.78 ACHE (0.52) TRPV1ACHEGRIN1GRIN2AGRIN2B
SCHEMBL2188030 0.78 ACHE (0.76) ACHEGRIN1GRIN2AGRIN2BGRIN2D
SCHEMBL21731608 0.77 MEN1 (0.55) HTR1ATRPV1DRD2DRD1DRD4
SCHEMBL3886166 0.77 BAZ2B (0.52) HTR1AACHEGRIN1GRIN2AGRIN2B
SCHEMBL25512689 0.77 L3MBTL1 (0.61) ACHEGRIN1GRIN2AGRIN2BGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed