SCHEMBL1662494

SCHEMBL1662494

CC(C)N(c1cc[nH]n1)c1nc(Cc2ccccc2C#N)c2cn[nH]c2n1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SGK1 O00141 1/20 0.34
EGFR P00533 1/20 0.32
PRKDC P78527 1/20 0.32
SLC5A1 P13866 1/20 0.31
SLC5A2 P31639 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801992 0.62 LRRK2 (0.37) SGK1HTR2AHTR2C
SCHEMBL28340016 0.58 CYP19A1 (0.41)
SCHEMBL27164099 0.57 SLC5A1 (0.38) SLC5A1SLC5A2
SCHEMBL11833453 0.56 CYP19A1 (0.39)
SCHEMBL2153612 0.56 CYP19A1 (0.48)
SCHEMBL27164207 0.56 ALDH1A1 (0.41)
SCHEMBL11837367 0.56 TSHR (0.41)
SCHEMBL11844643 0.56 IMPDH2 (0.41) HTR2AHTR2C
SCHEMBL27164067 0.55 TSHR (0.39) SLC5A1SLC5A2HTR2AHTR2C
SCHEMBL11840566 0.55 CYP19A1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2491039-A1 HETEROCYCLYL PYRAZOLOPYRIMIDINE ANALOGUES AS JAK INHIBITORS Cellzome Limited (GB) 2012-08-29 EP disclosed
WO-2011048082-A1 HETEROCYCLYL PYRAZOLOPYRIMIDINE ANALOGUES AS JAK INHIBITORS CELLZOME LIMITED (GB) 2011-04-28 WO disclosed