SCHEMBL1662613

SCHEMBL1662613

CC(C)(C)N1CCN(c2ccc(F)c(CO)c2F)CC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 3/20 0.34
TSHR P16473 2/20 0.34
POLB P06746 1/20 0.34
BRAF P15056 1/20 0.33
MAPK1 P28482 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PHGDH O43175 1/20 0.32
MAPT P10636 5/20 0.31
TDP1 Q9NUW8 2/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
LMNA P02545 1/20 0.31
GFER P55789 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663114 0.82 BRAF (0.31) ALDH1A1BRAFSMN1; SMN2
SCHEMBL28296311 0.81 PHGDH (0.40) ALDH1A1POLBMAPK1SMN1; SMN2PHGDH
SCHEMBL1662688 0.79 GPR119 (0.48) ALDH1A1SMN1; SMN2MAPTLMNAMEN1
SCHEMBL671924 0.77 AOC3 (0.38) ALDH1A1KDM4ETSHRPOLBMAPK1
SCHEMBL12631516 0.70 ALDH1A1 (0.46) ALDH1A1MAPK1SMN1; SMN2PHGDHMAPT
SCHEMBL12631522 0.69 SMN1; SMN2 (0.56) ALDH1A1KDM4ETSHRPOLBMAPK1
SCHEMBL27250548 0.68 ALDH1A1 (0.37) ALDH1A1KDM4ETSHRSMN1; SMN2MAPT
SCHEMBL16429868 0.68 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRPOLBMAPK1
SCHEMBL11364687 0.68 MAPT (0.60) ALDH1A1KDM4EPOLBMAPK1SMN1; SMN2
SCHEMBL671726 0.68 DRD2 (0.39) ALDH1A1KDM4ETSHRPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2491039-A1 HETEROCYCLYL PYRAZOLOPYRIMIDINE ANALOGUES AS JAK INHIBITORS Cellzome Limited (GB) 2012-08-29 EP disclosed
WO-2011048082-A1 HETEROCYCLYL PYRAZOLOPYRIMIDINE ANALOGUES AS JAK INHIBITORS CELLZOME LIMITED (GB) 2011-04-28 WO disclosed