SCHEMBL16626418

SCHEMBL16626418

CNCc1cn(S(=O)(=O)c2cccnc2)c2cc(Nc3ccc(F)cc3Cl)ccc12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.41
POLB P06746 2/20 0.38
FBP1 P09467 1/20 0.37
IDE P14735 2/20 0.36
HTR6 P50406 5/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
HTT P42858 2/20 0.35
MAP2K7 O14733 1/20 0.35
MAP2K4 P45985 1/20 0.35
TBXAS1 P24557 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16618755 0.99 NAMPT (0.40) NAMPTPOLBFBP1IDEHTR6
SCHEMBL16626428 0.92 HTR6 (0.41) NAMPTPOLBFBP1IDEHTR6
SCHEMBL17971520 0.92 POLB (0.42) NAMPTPOLBIDEHTR6HTT
Hydrochloric Acid SCHEMBL16618703 0.91 POLB (0.42) NAMPTPOLBIDEHTR6HTT
SCHEMBL16618670 0.91 NAMPT (0.41) NAMPTFBP1IDEHTR6PDE4A
SCHEMBL16626417 0.91 ALDH1A1 (0.40) NAMPTPOLBFBP1IDEHTR6
Hydrochloric Acid SCHEMBL16619520 0.91 HTR6 (0.40) NAMPTPOLBFBP1IDEHTR6
SCHEMBL16626431 0.90 NAMPT (0.38) NAMPTFBP1IDEHTR6PDE4A
SCHEMBL16626675 0.90 HTT (0.38) NAMPTFBP1IDEHTR6PDE4A
Hydrochloric Acid SCHEMBL16618639 0.90 ALDH1A1 (0.40) NAMPTPOLBFBP1IDEHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI NAMPT 1610/4885POLB 4594/4885FBP1 74/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.