SCHEMBL16626612

SCHEMBL16626612

CNCc1cn(S(=O)(=O)c2cccnc2)c2cc(Cc3ccc(C)nc3F)ccc12

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDE P14735 2/20 0.37
HTR6 P50406 7/20 0.36
ALK Q9UM73 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
TBXAS1 P24557 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
TSHR P16473 1/20 0.32
CYP19A1 P11511 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16618661 0.99 IDE (0.36) IDEHTR6ALKALDH1A1PDE4A
SCHEMBL16626626 0.90 IDE (0.37) IDEHTR6ALKPDE4APDE4B
Hydrochloric Acid SCHEMBL16619090 0.89 IDE (0.36) IDEHTR6ALKPDE4APDE4B
SCHEMBL16626654 0.87 IDE (0.37) IDEHTR6ALKALDH1A1PDE4A
SCHEMBL17971577 0.87 ALK (0.38) IDEHTR6ALKALDH1A1PDE4A
Hydrochloric Acid SCHEMBL16619344 0.86 ALK (0.38) IDEHTR6ALKALDH1A1PDE4A
Hydrochloric Acid SCHEMBL16619341 0.86 IDE (0.37) IDEHTR6ALKALDH1A1PDE4A
SCHEMBL16626640 0.86 HTR6 (0.40) IDEHTR6ALKALDH1A1TBXAS1
SCHEMBL17971580 0.85 ALK (0.41) IDEHTR6ALKPDE4APDE4B
Hydrochloric Acid SCHEMBL16619478 0.85 HTR6 (0.39) IDEHTR6ALKALDH1A1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI IDE 2586/4885HTR6 166/4885ALK 4825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.