SCHEMBL16627610

SCHEMBL16627610

C=Cc1ccc(N(C)C(=O)c2cc3c(NC(=O)/C=C/C)cccc3[nH]c2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 2/20 0.38
BTK Q06187 6/20 0.36
ALDH1A1 P00352 2/20 0.34
POLB P06746 2/20 0.34
KDM4E B2RXH2 3/20 0.32
NPC1 O15118 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
MAPT P10636 1/20 0.31
PELI1 Q96FA3 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC4 P56524 1/20 0.30
EP300 Q09472 1/20 0.30
MEF2D Q14814 1/20 0.30
PTGS2 P35354 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627614 0.89 PADI4 (0.39) PADI4BTKALDH1A1POLBKDM4E
SCHEMBL16627855 0.71 KDM4E (0.40) ALDH1A1KDM4EHSP90AA1HSP90AB1
SCHEMBL16627845 0.71 KDM4E (0.39) ALDH1A1POLBKDM4EMAPTHSP90AA1
SCHEMBL16627854 0.70 KDM4E (0.39) ALDH1A1KDM4ENPC1RXFP1HSP90AA1
SCHEMBL16627876 0.67 RXFP1 (0.44) POLBKDM4ENPC1RXFP1MAOB
SCHEMBL16627597 0.64 KMT2A (0.48) PADI4ALDH1A1KDM4ENPC1RXFP1
SCHEMBL16627896 0.63 PARP1 (0.40) ALDH1A1KDM4ENPC1RXFP1MAPT
SCHEMBL3644717 0.63 MAOB (0.56) PADI4ALDH1A1POLBKDM4EMAOB
SCHEMBL16627895 0.62 MEN1 (0.58) PADI4ALDH1A1KDM4ERXFP1MAOB
SCHEMBL16627787 0.62 PARP14 (0.47) ALDH1A1KDM4ENPC1RXFP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed