SCHEMBL16627614

SCHEMBL16627614

C/C=C/C(=O)Nc1cccc2[nH]c(=O)c(C(=O)N(C)c3ccc(O)cc3)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 1/20 0.39
BTK Q06187 5/20 0.38
HSP90AA1 P07900 4/20 0.36
PDK2 Q15119 2/20 0.36
PELI1 Q96FA3 1/20 0.36
PDK1 Q15118 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
MMP1 P03956 4/20 0.34
MMP2 P08253 4/20 0.34
MMP9 P14780 4/20 0.34
NPC1 O15118 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
HSP90AB1 P08238 2/20 0.33
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627610 0.89 PADI4 (0.38) PADI4BTKHSP90AA1PELI1KDM4E
SCHEMBL16627845 0.73 KDM4E (0.39) HSP90AA1KDM4EALDH1A1POLBMAPT
SCHEMBL16627855 0.73 KDM4E (0.40) HSP90AA1KDM4EALDH1A1HSP90AB1
SCHEMBL16627854 0.72 KDM4E (0.39) HSP90AA1KDM4EALDH1A1NPC1RXFP1
SCHEMBL16627680 0.71 PARP14 (0.48) HSP90AA1KDM4EALDH1A1HSP90AB1MEN1
SCHEMBL9182411 0.67 KDM4E (0.52) KDM4EALDH1A1POLBMAPTNPC1
SCHEMBL9302896 0.65 HSP90AA1 (0.46) HSP90AA1PDK2PDK1PDK3PDK4
SCHEMBL16627896 0.65 PARP1 (0.40) KDM4EALDH1A1MAPTNPC1RXFP1
SCHEMBL3644717 0.65 MAOB (0.56) PADI4KDM4EALDH1A1POLBMEN1
SCHEMBL16627895 0.64 MEN1 (0.58) PADI4KDM4EALDH1A1MAPTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed