SCHEMBL16627616

SCHEMBL16627616

CCNC(=O)c1cc2c(NC(=O)c3ccccc3)cccc2[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.53
KDM4E B2RXH2 3/20 0.49
PARP14 Q460N5 1/20 0.47
BRD4 O60885 1/20 0.46
BACE1 P56817 1/20 0.45
NPC1 O15118 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
STK33 Q9BYT3 1/20 0.45
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
PSMB8 P28062 1/20 0.44
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627785 0.87 TOP1 (0.48) PARP1KDM4EPARP14NPC1RAB9A
SCHEMBL16627819 0.85 BRD4 (0.54) PARP1PARP14BRD4NPC1CYP1A2
SCHEMBL16627818 0.78 RXFP1 (0.53) PARP1BRD4NPC1RAB9AMAPT
SCHEMBL16627598 0.75 SMYD3 (0.54) KDM4EBRD4ALDH1A1TSHRHSD17B10
SCHEMBL10813245 0.72 PARP1 (0.57) PARP1KDM4EPARP14BRD4NPC1
SCHEMBL16627806 0.72 NHERF1 (0.49) PARP1KDM4ESTK33MAPTALDH1A1
SCHEMBL16627879 0.71 MAPT (0.51) PARP1KDM4ENPC1RAB9ASTK33
SCHEMBL16627787 0.70 PARP14 (0.47) KDM4EPARP14NPC1CYP2C9RAB9A
SCHEMBL16627688 0.70 MAPT (0.50) KDM4ENPC1RAB9AMAPTALDH1A1
SCHEMBL16627783 0.70 PARP14 (0.47) KDM4EPARP14NPC1CYP2C9RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed