SCHEMBL16627762

SCHEMBL16627762

C=Cc1ccc(NC(=O)c2cc3ccccc3n(CC)c2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.56
MAPT P10636 3/20 0.47
TP53 P04637 1/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
CNR1 P21554 6/20 0.45
CNR2 P34972 5/20 0.45
MAOB P27338 2/20 0.45
POLB P06746 2/20 0.44
MAPK1 P28482 2/20 0.44
BLM P54132 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.43
MAOA P21397 1/20 0.42
NPC1 O15118 1/20 0.42
APOBEC3A P31941 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627741 0.89 AHR (0.61) AHRMAPTTP53MEN1KMT2A
SCHEMBL16627748 0.87 AHR (0.73) AHRMAPTTP53MEN1KMT2A
SCHEMBL16627757 0.86 AHR (0.72) AHRMAPTTP53MEN1KMT2A
SCHEMBL16627658 0.81 CNR1 (0.50) AHRCNR1CNR2
SCHEMBL16627568 0.76 CA12 (0.51) CNR1CNR2POLBMAPK1ALDH1A1
SCHEMBL16627681 0.75 NPY5R (0.45) MAPTMEN1KMT2APOLBMAPK1
SCHEMBL30237030 0.74 AHR (0.85) AHRMEN1KMT2AMAOBPOLB
SCHEMBL1397253 0.74 AHR (0.85) AHRMEN1KMT2AMAOBPOLB
SCHEMBL6547150 0.73 MAPK1 (0.47) KMT2ACNR1CNR2MAPK1ALDH1A1
SCHEMBL16627765 0.73 MAPK1 (0.47) MAPTTP53CNR1CNR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed