SCHEMBL16629085

SCHEMBL16629085

NC(=O)Nc1ccc(CN2CCC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
TNIK Q9UKE5 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.58
HRH3 Q9Y5N1 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.53
GAA P10253 2/20 0.52
TNF P01375 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 2/20 0.51
TP53 P04637 1/20 0.51
POLB P06746 1/20 0.51
CHRM1 P11229 2/20 0.51
HTR2A P28223 2/20 0.51
MCHR1 Q99705 2/20 0.51
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9035239 0.95 KDM4E (0.72) KDM4EALDH1A1TNIKL3MBTL1HRH3
SCHEMBL18925150 0.86 HDAC6 (0.58) KDM4EALDH1A1TNIKSMN1; SMN2GAA
SCHEMBL30486118 0.86 RAB9A (0.70) KDM4EALDH1A1TNIKL3MBTL1SMN1; SMN2
SCHEMBL30860319 0.83 ALDH1A1 (0.54) KDM4EALDH1A1TNIKL3MBTL1HRH3
SCHEMBL15156423 0.79 KDM4E (1.00) KDM4EALDH1A1TNIKL3MBTL1HRH3
SCHEMBL10515943 0.78 CDK5 (0.56) ALDH1A1SMN1; SMN2POLBCHEK1
SCHEMBL6224393 0.77 HRH3 (0.55) KDM4EALDH1A1L3MBTL1HRH3SMN1; SMN2
SCHEMBL7008043 0.75 KDM4E (0.67) KDM4EALDH1A1TNIKL3MBTL1HRH3
SCHEMBL25230264 0.74 NPC1 (0.61) ALDH1A1GAANPC1LMNAKMT2A
SCHEMBL694950 0.74 RAB9A (0.73) KDM4EALDH1A1L3MBTL1HRH3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049325-A1 THERAPEUTIC INHIBITORS OF CDK8 AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2015-04-09 WO disclosed