SCHEMBL7008043

SCHEMBL7008043

O=C(Nc1ccc(CN2CCCCC2)cc1)C(F)(F)F

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.67
ALDH1A1 P00352 2/20 0.67
TNIK Q9UKE5 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
MCHR1 Q99705 3/20 0.55
HRH3 Q9Y5N1 2/20 0.54
GAA P10253 3/20 0.54
TNF P01375 1/20 0.54
CHRM1 P11229 2/20 0.53
HTR2A P28223 2/20 0.53
LMNA P02545 1/20 0.53
KMT2A Q03164 1/20 0.53
HTT P42858 1/20 0.53
RAB9A P51151 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9035239 0.80 KDM4E (0.72) KDM4EALDH1A1TNIKL3MBTL1SMN1; SMN2
SCHEMBL15156423 0.80 KDM4E (1.00) KDM4EALDH1A1TNIKL3MBTL1SMN1; SMN2
SCHEMBL3166509 0.79 KIT (0.51) SMN1; SMN2
SCHEMBL1604864 0.76 KDM4E (0.66) KDM4EALDH1A1TNIKL3MBTL1SMN1; SMN2
SCHEMBL11077344 0.76 CA12 (0.56) L3MBTL1SMN1; SMN2GAALMNAKMT2A
SCHEMBL694950 0.75 RAB9A (0.73) KDM4EALDH1A1L3MBTL1SMN1; SMN2HRH3
SCHEMBL16629085 0.75 KDM4E (0.65) KDM4EALDH1A1TNIKL3MBTL1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL2269036 0.75 ALDH1A1 (0.57) KDM4EALDH1A1HRH3GAALMNA
SCHEMBL16620534 0.75 KDM4E (0.48) KDM4EALDH1A1SMN1; SMN2HRH3GAA
SCHEMBL28663251 0.74 RAB9A (0.76) KDM4EALDH1A1L3MBTL1MCHR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1315726-A1 7- OXO PYRIDOPYRIMIDINES AS INHIBITORS OF CELLULAR PROLIFERATION F. HOFFMANN-LA ROCHE AG (CH) 2003-06-04 EP disclosed
WO-2002018380-A1 7-OXO PYRIDOPYRIMIDINES AS INHIBITORS OF A CELLULAR PROLIFERATION F. HOFFMANN-LA ROCHE AG (CH) 2002-03-07 WO disclosed