SCHEMBL9035239

SCHEMBL9035239

NC(=O)Nc1ccc(CN2CCCCC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.72
ALDH1A1 P00352 1/20 0.72
L3MBTL1 Q9Y468 1/20 0.64
TNIK Q9UKE5 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.59
HRH3 Q9Y5N1 2/20 0.58
GAA P10253 3/20 0.58
TNF P01375 1/20 0.58
MCHR1 Q99705 3/20 0.56
CHRM1 P11229 2/20 0.56
HTR2A P28223 2/20 0.56
LMNA P02545 1/20 0.56
KMT2A Q03164 1/20 0.56
HTT P42858 1/20 0.56
RAB9A P51151 1/20 0.56
CHEK1 O14757 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16629085 0.95 KDM4E (0.65) KDM4EALDH1A1L3MBTL1TNIKSMN1; SMN2
SCHEMBL30486118 0.84 RAB9A (0.70) KDM4EALDH1A1L3MBTL1TNIKSMN1; SMN2
SCHEMBL18925150 0.84 HDAC6 (0.58) KDM4EALDH1A1TNIKSMN1; SMN2GAA
SCHEMBL15156423 0.84 KDM4E (1.00) KDM4EALDH1A1L3MBTL1TNIKSMN1; SMN2
SCHEMBL30860319 0.82 ALDH1A1 (0.54) KDM4EALDH1A1L3MBTL1TNIKSMN1; SMN2
SCHEMBL7008043 0.80 KDM4E (0.67) KDM4EALDH1A1L3MBTL1TNIKSMN1; SMN2
SCHEMBL10515943 0.80 CDK5 (0.56) ALDH1A1SMN1; SMN2CHEK1
SCHEMBL28247816 0.80 TNF (0.71) KDM4EALDH1A1L3MBTL1SMN1; SMN2GAA
SCHEMBL694950 0.79 RAB9A (0.73) KDM4EALDH1A1L3MBTL1SMN1; SMN2HRH3
SCHEMBL2912150 0.78 HRH3 (0.64) KDM4EALDH1A1HRH3GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0719264-A1 IMIDAZOLONE AND OXAZOLONE DERIVATIVES AS DOPAMINE ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1996-07-03 EP disclosed
WO-1995007904-A1 IMIDAZOLONE AND OXAZOLONE DERIVATIVES AS DOPAMINE ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-03-23 WO disclosed