SCHEMBL16629591

SCHEMBL16629591

CC(C)Cc1cccc(-c2ccc3c(c2)OCO3)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.56
SLC6A4 P31645 3/20 0.56
SLC6A2 P23975 2/20 0.56
SLC6A3 Q01959 2/20 0.56
GABRA1 P14867 1/20 0.51
GABRB2 P47870 1/20 0.51
CYP2D6 P10635 2/20 0.50
NPSR1 Q6W5P4 1/20 0.46
PTPRC P08575 1/20 0.46
CYP3A4 P08684 2/20 0.45
FYN P06241 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CALM1 P0DP23 1/20 0.43
PTGS2 P35354 1/20 0.43
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18015825 0.83 MAPT (0.55) TAAR1SLC6A4SLC6A2SLC6A3GABRA1
SCHEMBL104467 0.82 TAAR1 (0.74) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL28161128 0.80 CTSS (0.48) TAAR1SLC6A4SLC6A2SLC6A3GABRA1
SCHEMBL16675752 0.80 FYN (0.59) GABRA1GABRB2CYP2D6PTPRCCYP3A4
SCHEMBL2929152 0.80 CALM1 (0.46) GABRA1GABRB2CYP2D6PTPRCCYP3A4
SCHEMBL18014706 0.79 GABRA1 (0.45) TAAR1SLC6A4SLC6A2SLC6A3GABRA1
SCHEMBL2692579 0.78 CA12 (0.59) GABRA1GABRB2PTPRCCYP3A4NPC1
SCHEMBL29629010 0.78 PTGS2 (0.58) GABRA1GABRB2PTPRCCYP3A4NPC1
SCHEMBL8636391 0.77 MEN1 (0.46) TAAR1SLC6A4SLC6A2SLC6A3GABRA1
SCHEMBL14200080 0.76 GABRA1 (0.55) TAAR1SLC6A4SLC6A2SLC6A3GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049616-A1 NOVEL BICYCLIC PYRIDINONES AS GAMMA-SECRETASE MODULATORS PFIZER INC. (US) 2015-04-09 WO disclosed