SCHEMBL16630218

SCHEMBL16630218

CN(Cc1cncc(F)c1)C(=O)c1ccc(C[C@@H]2CC[C@H]([C@H](O)c3ccccc3)N2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CETP P11597 5/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GPR119 Q8TDV5 1/20 0.34
LIMK2 P53671 1/20 0.34
JAK2 O60674 1/20 0.33
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33
USP30 Q70CQ3 1/20 0.33
CCR5 P51681 1/20 0.33
TACR1 P25103 1/20 0.33
NAMPT P43490 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
USP1 O94782 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16629828 0.91 CETP (0.38) CETPMEN1KMT2AGPR119LIMK2
SCHEMBL16629823 0.90 CETP (0.36) CETPMEN1KMT2AGPR119LIMK2
SCHEMBL16629855 0.89 GPR119 (0.42) CETPMEN1KMT2AGPR119LIMK2
SCHEMBL18017460 0.89 CETP (0.34) CETPMEN1KMT2AGPR119LIMK2
SCHEMBL16629921 0.88 CETP (0.38) CETPMEN1KMT2AGPR119LIMK2
SCHEMBL21278650 0.86 GPR119 (0.41) CETPGPR119LIMK2USP30
SCHEMBL16630588 0.85 ACACB (0.40) MEN1KMT2AGPR119
SCHEMBL18017442 0.83 ACACB (0.41) MEN1KMT2AGPR119USP30NAMPT
SCHEMBL21278623 0.82 GRM5 (0.42) CETPMEN1KMT2AGPR119JAK2
SCHEMBL31012162 0.81 CETP (0.40) CETPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed