SCHEMBL16629823

SCHEMBL16629823

COC(=O)c1cncc(CN(C)C(=O)c2ccc(C[C@@H]3CC[C@H]([C@H](O)c4ccccc4)N3C(=O)OC(C)(C)C)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.36
LIMK2 P53671 1/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34
GPR119 Q8TDV5 2/20 0.33
SLC2A1 P11166 1/20 0.33
CCR5 P51681 1/20 0.33
JAK2 O60674 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
USP30 Q70CQ3 1/20 0.32
ACKR3 P25106 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16630218 0.90 CETP (0.37) CETPLIMK2ABL1RIN1GPR119
SCHEMBL16629828 0.89 CETP (0.38) CETPLIMK2ABL1RIN1GPR119
SCHEMBL18017455 0.89 CETP (0.34) CETPLIMK2HDAC1HDAC6ABL1
SCHEMBL16630680 0.89 CETP (0.34) CETPLIMK2HDAC1HDAC6ABL1
SCHEMBL16629855 0.88 GPR119 (0.42) CETPLIMK2GPR119SLC2A1MEN1
SCHEMBL21278650 0.84 GPR119 (0.41) CETPLIMK2GPR119USP30
SCHEMBL16629921 0.84 CETP (0.38) CETPLIMK2HDAC1ABL1RIN1
SCHEMBL16630588 0.84 ACACB (0.40) GPR119MEN1KMT2A
SCHEMBL16629922 0.83 P2RX3 (0.34) HDAC1HDAC6GPR119
SCHEMBL17986551 0.82 LIMK2 (0.33) CETPLIMK2ABL1RIN1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed