SCHEMBL16630760

SCHEMBL16630760

Cc1nnc2ccc(CN(C)C(=O)c3ccc(C[C@@H]4CC[C@H]([C@H](O)c5ccc(Cl)nc5)N4C(=O)OC(C)(C)C)cc3)cn12

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.31
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
CETP P11597 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18017468 0.90
SCHEMBL16629834 0.89 AGTR2 (0.36) GPR119CETP
SCHEMBL21278147 0.84 CETP (0.34) GPR119CETP
SCHEMBL18017457 0.82 MAPK14 (0.39) GPR119CETP
SCHEMBL16620038 0.81 ADRB1 (0.38) GPR119CETP
SCHEMBL18017379 0.81 ADRB1 (0.38) GPR119CETP
SCHEMBL16620041 0.81 ADRB1 (0.38) GPR119CETP
SCHEMBL16619851 0.79 ADRB3 (0.38)
SCHEMBL16619853 0.79 ADRB3 (0.38)
SCHEMBL21278412 0.79 GPR119 (0.36) GPR119CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed