SCHEMBL16629834

SCHEMBL16629834

CN(Cc1ccc(Cl)nc1)C(=O)c1ccc(C[C@@H]2CC[C@H]([C@H](O)c3ccc(Cl)nc3)N2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.36
GPR119 Q8TDV5 11/20 0.35
CETP P11597 4/20 0.34
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21278147 0.92 CETP (0.34) AGTR2GPR119CETP
SCHEMBL16630760 0.89 GPR119 (0.31) GPR119CETP
SCHEMBL18017452 0.88 AGTR2 (0.33) AGTR2GPR119CETP
SCHEMBL16620041 0.88 ADRB1 (0.38) GPR119CETPCHRNB2CHRNA7CHRNA4
SCHEMBL18017379 0.88 ADRB1 (0.38) GPR119CETPCHRNB2CHRNA7CHRNA4
SCHEMBL16620038 0.88 ADRB1 (0.38) GPR119CETPCHRNB2CHRNA7CHRNA4
SCHEMBL21278412 0.87 GPR119 (0.36) GPR119CETPCHRNB2CHRNA7CHRNA4
SCHEMBL18017457 0.86 MAPK14 (0.39) GPR119CETPCHRNB2CHRNA4
SCHEMBL16629887 0.85 GPR119 (0.37) GPR119CETPKMT2A
SCHEMBL18210822 0.85 ACKR3 (0.38) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed